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Sodium channel
protein type 10
subunit alpha
Sodium channel
subunit beta-1
Cytochrome P450
1A2
Cytochrome P450
3A4
Cytochrome P450
1A2
Cytochrome P450
3A4
Lidocaine
Lidocaine
2,6-Dimethylaniline
Monoethylglycinexylidide
Glycinexylidide
2-Amino-3-methylbenzoate
4-Hydroxy-2,6-dimethylaniline
3-Hydroxylidocaine
3-
Hydroxymonoethylglycinexylidide
O
2
NADPH
H
+
H
2
O
NADP
O
2
NADH
H
2
O
Formaldehyde
NAD
Heme
Heme
Heme
Heme
Axon
Voltage-gated sodium channel
(INa)
SCN10A
SCN1B
CYP1A2
CYP3A4
CYP1A2
CYP3A4
Lidocaine
Lidocaine
2,6-
Dimethylaniline
Monoethylglycinexylidide
Glycinexylidide
2-Amino-3-
methylbenzoate
4-Hydroxy- 2,6-
dimethylaniline
3-
Hydroxylidocaine
3-
Hydroxymonoethylglycinexylidide
Oxygen
NADPH
Hydrogen Ion
Water
NADP
Oxygen
NADH
Water
Formaldehyde
NAD
SCN10A
SCN1B
CYP1A2
CYP3A4
CYP1A2
CYP3A4
L-Caine
L-Caine
2,6-Dma
Monoeg
Glycxyl
2A3M
4H26MAl
3-HLido
3-HMegc
O
2
NADPH
H
+
H
2
O
NADP
O
2
NADH
H
2
O
Formol
NAD
Heme
Heme
Heme
Heme