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Cytochrome P450 3A4 Alectinib Alectinib Alectinib PIS1M1 Alectinib PIS1M1 Urinary Excretion and/or Bile duct Excretion Heme Hepatocytes Kidney Liver Cytosol Alectinib undergoes metabolism to give Alectinib PIS1M1. Endoplasmic Reticulum Bile Ducts Blood Vessel Blood Vessel
Endoplasmic Reticulum CYP3A4 Alectinib Alectinib Alectinib PIS1M1 Alectinib PIS1M1 Urinary Excretion and/or Bile duct Excretion
CYP3A4 Alect Alect Ale PIS Ale PIS U E a B Heme Hepatocytes Kidney Liver Cytosol Alectinib undergoes metabolism to give Alectinib PIS1M1. Endoplasmic Reticulum Bile Ducts Blood Vessel Blood Vessel
Endoplasmic Reticulum CYP3A4 Alect Alect Ale PIS Ale PIS U E a B