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Unknown Unknown Unknown Cytochrome P450 3A4 Cytochrome P450 3A4 Cytochrome P450 3A4 Alosetron Alosetron Alosetron PIS1M2 Alosetron PIS2M1 Alosetron PIS2M1 Alosetron PIS1M1 Alosetron PIS1M2 Heme Heme Heme Urinary Excretion and/or Bile duct Excretion Endoplasmic Reticulum Cytosol Hepatocyte Blood Vessel Liver kidney Bile Duct Blood Vessel Alosetron undergoes metabolism to give Alosetron PIS1M1, Alosetron PIS1M2 and Alosetron PIS2M1. Endoplasmic Reticulum
Endoplasmic Reticulum Endoplasmic Reticulum Unknown Unknown Unknown CYP3A4 CYP3A4 CYP3A4 Alosetron Alosetron Alosetron PIS1M2 Alosetron PIS2M1 Alosetron PIS2M1 Alosetron PIS1M1 Alosetron PIS1M2 Urinary Excretion and/or Bile duct Excretion