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Unknown Unknown Unknown Cytochrome P450 3A4 Cytochrome P450 3A4 Cytochrome P450 3A4 Cilostazol Cilostazol Cilostazol PIS1M2 Cilostazol PIS2M1 Cilostazol PIS2M1 Cilostazol PIS1M1 Cilostazol PIS1M2 Heme Heme Heme Urinary Excretion and/or Bile duct Excretion Endoplasmic Reticulum Cytosol Hepatocyte Blood Vessel Liver kidney Bile Duct Blood Vessel Cilostazol undergoes metabolism to give Cilostazol PIS1M1, Cilostazol PIS1M2 and Cilostazol PIS2M1. Endoplasmic Reticulum
Endoplasmic Reticulum Endoplasmic Reticulum Unknown Unknown Unknown CYP3A4 CYP3A4 CYP3A4 Cilostazol Cilostazol Cilostazol PIS1M2 Cilostazol PIS2M1 Cilostazol PIS2M1 Cilostazol PIS1M1 Cilostazol PIS1M2 Urinary Excretion and/or Bile duct Excretion